平安! 发表于 2011-11-9 19:57 7 [" ]6 c/ s6 C! `9 R
Pazopanib (100 mg/kg/day free base equivalent)
2 V( h3 n6 k- z: D, u8 m 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。. L0 \. U# ?, r. w
搜索了一下,原料一大堆。) S+ R' p, C* n5 T
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对不起!100mg/kg是用于移植瘤的,我弄错了。/ {' n! W. w1 i% G) C+ `% ]8 O/ S
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以下是正版说明书的推荐用量。( O0 W2 k) l8 \# i, h
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--------------------- DOSAGE AND ADMINISTRATION ----------------
2 A+ C6 v5 ^3 o* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) ' i( C* B* `% P, X9 \
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
) P5 D+ c& i6 y* h5 |' w. a---------------------DOSAGE FORMS AND STRENGTHS --------------
) t3 H) ~# z( k1 C$ Z" F3 C0 A200 mg tablets. (3) 9 ]9 Q0 k& N/ o( A6 t; \
-------------------------------CONTRAINDICATIONS------------------------ |